{"id":9093,"date":"2019-02-28T20:42:00","date_gmt":"2019-02-28T20:42:00","guid":{"rendered":"https:\/\/dupmecp2.eu\/drug-repositioning-study-at-apteeus\/"},"modified":"2022-11-11T19:36:12","modified_gmt":"2022-11-11T19:36:12","slug":"drug-repositioning-study-at-apteeus","status":"publish","type":"post","link":"https:\/\/dupmecp2.eu\/en\/drug-repositioning-study-at-apteeus\/","title":{"rendered":"Drug repositioning study at APTEEUS\u2122"},"content":{"rendered":"<p class=\"has-text-align-left\">The first phase of the project conducted by APTEEUS\u2122 with Les petits Mec P2 Association is coming to an end. Duplication of the MECP2 gene results in overexpression of the MeCP2 protein present in all cells of the body. APTEEUS\u2122 chose to use fibroblasts from the patients' skin to highlight the overexpression of the protein and attempt to regulate it with molecules already used for other indications. <\/p>\n\n<p class=\"has-text-align-left\">Among more than 5,000 molecules tested during the screening, APTEEUS\u2122 has identified several molecules capable of reducing the amount of MeCP2 protein in the cells of 2 patients in the association. <\/p>\n\n<p class=\"has-text-align-left\">APTEEUS\u2122 is currently collecting data on each of the selected molecules so that we can judge their medical interest with physicians.<br\/><\/p>\n\n<figure class=\"wp-block-image size-large\"><img fetchpriority=\"high\" decoding=\"async\" width=\"1024\" height=\"561\" src=\"https:\/\/dupmecp2.eu\/wp-content\/uploads\/2022\/07\/illustrationcriblage-1400x767-1-1024x561.png\" alt=\"\" class=\"wp-image-3101\" srcset=\"https:\/\/dupmecp2.eu\/wp-content\/uploads\/2022\/07\/illustrationcriblage-1400x767-1-1024x561.png 1024w, https:\/\/dupmecp2.eu\/wp-content\/uploads\/2022\/07\/illustrationcriblage-1400x767-1-300x164.png 300w, https:\/\/dupmecp2.eu\/wp-content\/uploads\/2022\/07\/illustrationcriblage-1400x767-1-768x421.png 768w, https:\/\/dupmecp2.eu\/wp-content\/uploads\/2022\/07\/illustrationcriblage-1400x767-1-600x329.png 600w, https:\/\/dupmecp2.eu\/wp-content\/uploads\/2022\/07\/illustrationcriblage-1400x767-1.png 1400w\" sizes=\"(max-width: 1024px) 100vw, 1024px\" \/><figcaption class=\"wp-element-caption\">Illustration of screening results. The control level of MeCP2 is normally less than 6.0.10<sup>5<\/sup>, whereas the patient cells have a level close to 1,0.10<sup>6<\/sup>.<\/figcaption><\/figure>\n\n<p><\/p>","protected":false},"excerpt":{"rendered":"<p>The first phase of the project conducted by APTEEUS&#x2122; with Les petits Mec P2 Association is coming to an end. Duplication of the MECP2 gene results in overexpression of the [&hellip;]<\/p>","protected":false},"author":1,"featured_media":3102,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[87],"tags":[],"class_list":["post-9093","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-news"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v25.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Drug repositioning study at APTEEUS&#x2122; - DupMECP2<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/dupmecp2.eu\/en\/drug-repositioning-study-at-apteeus\/?lang=en\" \/>\n<meta property=\"og:locale\" content=\"en_GB\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Drug repositioning study at APTEEUS&#x2122; - DupMECP2\" \/>\n<meta property=\"og:description\" content=\"The first phase of the project conducted by APTEEUS&#x2122; with Les petits Mec P2 Association is coming to an end. Duplication of the MECP2 gene results in overexpression of the [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/dupmecp2.eu\/en\/drug-repositioning-study-at-apteeus\/?lang=en\" \/>\n<meta property=\"og:site_name\" content=\"DupMECP2\" \/>\n<meta property=\"article:published_time\" content=\"2019-02-28T20:42:00+00:00\" \/>\n<meta property=\"article:modified_time\" content=\"2022-11-11T19:36:12+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/dupmecp2.eu\/wp-content\/uploads\/2022\/07\/illustrationcriblage-1400x767-1.png\" \/>\n\t<meta property=\"og:image:width\" content=\"1400\" \/>\n\t<meta property=\"og:image:height\" content=\"767\" \/>\n\t<meta property=\"og:image:type\" content=\"image\/png\" \/>\n<meta name=\"author\" content=\"Caroline\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Written by\" \/>\n\t<meta name=\"twitter:data1\" content=\"Caroline\" \/>\n\t<meta name=\"twitter:label2\" content=\"Estimated reading time\" \/>\n\t<meta name=\"twitter:data2\" content=\"1 minute\" \/>\n<script type=\"application\/ld+json\" class=\"yoast-schema-graph\">{\"@context\":\"https:\/\/schema.org\",\"@graph\":[{\"@type\":\"Article\",\"@id\":\"https:\/\/dupmecp2.eu\/drug-repositioning-study-at-apteeus\/?lang=en#article\",\"isPartOf\":{\"@id\":\"https:\/\/dupmecp2.eu\/drug-repositioning-study-at-apteeus\/?lang=en\"},\"author\":{\"name\":\"Caroline\",\"@id\":\"https:\/\/dupmecp2.eu\/#\/schema\/person\/b41e8cbba153cd974ee340386af279ee\"},\"headline\":\"Drug repositioning study at APTEEUS&#x2122;\",\"datePublished\":\"2019-02-28T20:42:00+00:00\",\"dateModified\":\"2022-11-11T19:36:12+00:00\",\"mainEntityOfPage\":{\"@id\":\"https:\/\/dupmecp2.eu\/drug-repositioning-study-at-apteeus\/?lang=en\"},\"wordCount\":149,\"publisher\":{\"@id\":\"https:\/\/dupmecp2.eu\/#organization\"},\"image\":{\"@id\":\"https:\/\/dupmecp2.eu\/drug-repositioning-study-at-apteeus\/?lang=en#primaryimage\"},\"thumbnailUrl\":\"https:\/\/dupmecp2.eu\/wp-content\/uploads\/2022\/07\/illustrationcriblage-1400x767-1.png\",\"articleSection\":[\"News\"],\"inLanguage\":\"en-GB\"},{\"@type\":\"WebPage\",\"@id\":\"https:\/\/dupmecp2.eu\/drug-repositioning-study-at-apteeus\/?lang=en\",\"url\":\"https:\/\/dupmecp2.eu\/drug-repositioning-study-at-apteeus\/?lang=en\",\"name\":\"Drug repositioning study at APTEEUS&#x2122; 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